Bourdonnec, Bertrand Le: search on Z-Library

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1

ChemInform Abstract: Pyrazolidine-3,5-dione Angiotensin-II Receptor Antagonists

Christine Cauvin, Bertrand Le Bourdonnec, Bernadette Norberg, Jean-Pierre Henichart, Francois Durant

Journal:

Year:

2002

File:

PDF, 28 KB

2002

2

ChemInform Abstract: Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2008

Roland E. Dolle, Bertrand Le Bourdonnec, Allan J. Goodman, Guillermo A. Morales, Craig J. Thomas, Wei Zhang

Journal:

Year:

2010

File:

PDF, 16 KB

2010

3

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2007

Dolle, Roland E., Bourdonnec, Bertrand Le, Goodman, Allan J., Morales, Guillermo A., Thomas, Craig J., Zhang, Wei

Journal:

Journal of Combinatorial Chemistry

Year:

2008

Language:

english

File:

PDF, 5.69 MB

english, 2008

4

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2009

Dolle, Roland E., Bourdonnec, Bertrand Le, Worm, Karin, Morales, Guillermo A., Thomas, Craig J., Zhang, Wei

Journal:

Journal of Combinatorial Chemistry

Year:

2010

Language:

english

File:

PDF, 2.85 MB

english, 2010

5

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2008

Dolle, Roland E., Bourdonnec, Bertrand Le, Goodman, Allan J., Morales, Guillermo A., Thomas, Craig J., Zhang, Wei

Journal:

Journal of Combinatorial Chemistry

Year:

2009

Language:

english

File:

PDF, 10.29 MB

english, 2009

6

Synthesis and structure–activity relationships of a new series of 2α-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as μ-selective opioid antagonists

Bertrand Le Bourdonnec, Allan J. Goodman, Mathieu Michaut, Hai-Fen Ye, Thomas M. Graczyk, Serge Belanger, Robert N. DeHaven, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 198 KB

english, 2006

7

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2006

Dolle, Roland E., Le Bourdonnec, Bertrand, Goodman, Allan J., Morales, Guillermo A., Salvino, Joseph M., Zhang, Wei

Journal:

Journal of Combinatorial Chemistry

Year:

2007

Language:

english

File:

PDF, 5.14 MB

english, 2007

8

Comprehensive Survey of Combinatorial Library Synthesis: 2005

Dolle, Roland E., Le Bourdonnec, Bertrand, Morales, Guillermo A., Moriarty, Kevin J., Salvino, Joseph M.

Journal:

Journal of Combinatorial Chemistry

Year:

2006

Language:

english

File:

PDF, 3.49 MB

english, 2006

9

A new synthesis of N-alkyl pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones

Bertrand Le Bourdonnec, Emmanuelle Meulon, Saïd Yous, Raymond Houssin, Jean-Pierre Hénichart

Journal:

Journal of Heterocyclic Chemistry

Year:

2000

File:

PDF, 335 KB

2000

10

Potent, Orally Bioavailable Delta Opioid Receptor Agonists for the Treatment of Pain: Discovery of N , N -Diethyl-4-(5-hydroxyspiro[chromene-2,4′-piperidine]-4-yl)benzamide (ADL5859)

Bourdonnec, Bertrand Le, Windh, Rolf T., Ajello, Christopher W., Leister, Lara K., Gu, Minghua, Chu, Guo-Hua, Tuthill, Paul A., Barker, William M., Koblish, Michael, Wiant, Daniel D., Graczyk, Thomas

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 125 KB

english, 2008

11

Mu Opioid Receptor Antagonists: Recent Developments

Allan J. Goodman, Bertrand Le Bourdonnec, Roland E. Dolle

Journal:

Year:

2007

Language:

english

File:

PDF, 804 KB

english, 2007

12

trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of μ-Selective opioid antagonists

Bertrand Le Bourdonnec, Serge Belanger, Joel A. Cassel, Gabriel J. Stabley, Robert N. DeHaven, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 198 KB

english, 2003

13

Discovery of a series of aminopiperidines as novel iNOS inhibitors

Bertrand Le Bourdonnec, Lara K. Leister, Christopher A. Ajello, Joel A. Cassel, Pamela R. Seida, Heather O’Hare, Minghua Gu, Guo-Hua Chu, Paul A. Tuthill, Robert N. DeHaven, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 294 KB

english, 2008

14

Synthesis and Pharmacological Evaluation of New Pyrazolidine-3,5-diones as AT 1 Angiotensin II Receptor Antagonists

Le Bourdonnec, Bertrand, Meulon, Emmanuelle, Yous, Saïd, Goossens, Jean-François, Houssin, Raymond, Hénichart, Jean-Pierre

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 179 KB

english, 2000

15

Naphthalene Dicarboxaldehyde as an Electrophilic Fluorogenic Moiety for Affinity Labeling: Application to Opioid Receptor Affinity Labels with Greatly Improved Fluorogenic Properties

McCurdy, Christopher R., Le Bourdonnec, Bertrand, Metzger, Thomas G., El Kouhen, Rachid, Zhang, Yan, Law, Ping Y., Portoghese, Philip S.

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 71 KB

english, 2002

16

ChemInform Abstract: Affinity Labels as Tools for the Identification of Opioid Receptor Recognition Sites

Philip S. Portoghese, Rachid El Kouhen, Ping Y. Law, Horace H. Loh, Bertrand Le Bourdonnec

Journal:

Year:

2001

File:

PDF, 26 KB

2001

17

Arylacetamide κ opioid receptor agonists with reduced cytochrome P450 2D6 inhibitory activity

Bertrand Le Bourdonnec, Christopher W. Ajello, Pamela R. Seida, Roberta G. Susnow, Joel A. Cassel, Serge Belanger, Gabriel J. Stabley, Robert N. DeHaven, Diane L. DeHaven-Hudkins, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 182 KB

english, 2005

18

o -Naphthalenedicarboxaldehyde Derivative of 7‘-Aminonaltrindole as a Selective δ-Opioid Receptor Affinity Label

Haris, Sarika Prabhu, Zhang, Yan, Le Bourdonnec, Bertrand, McCurdy, Christopher R., Portoghese, Philip S.

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 116 KB

english, 2007

19

Spirocyclic Delta Opioid Receptor Agonists for the Treatment of Pain: Discovery of N , N -Diethyl-3-hydroxy-4-(spiro[chromene-2,4′-piperidine]-4-yl) Benzamide (ADL5747)

Le Bourdonnec, Bertrand, Windh, Rolf T., Leister, Lara K., Zhou, Q. Jean, Ajello, Christopher W., Gu, Minghua, Chu, Guo-Hua, Tuthill, Paul A., Barker, William M., Koblish, Michael, Wiant, Daniel D., G

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 1.65 MB

english, 2009

20

Covalently Induced Activation of the δ Opioid Receptor by a Fluorogenic Affinity Label, 7‘-(Phthalaldehydecarboxamido)naltrindole (PNTI)

Le Bourdonnec, Bertrand, El Kouhen, Rachid, Poda, Gennady, Law, Ping Y., Loh, Horace H., Ferguson, David M., Portoghese, Philip S.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 185 KB

english, 2001

21

Elucidation of the Bioactive Conformation of the N -Substituted trans -3,4-Dimethyl-4-(3-hydroxyphenyl)piperidine Class of μ-Opioid Receptor Antagonists

Le Bourdonnec, Bertrand, Goodman, Allan J., Michaut, Mathieu, Ye, Hai-Fen, Graczyk, Thomas M., Belanger, Serge, Herbertz, Torsten, Yap, Glenn P. A., DeHaven, Robert N., Dolle, Roland E.

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 223 KB

english, 2006

22

Novel sulfamoyl benzamides as selective CB2 agonists with improved in vitro metabolic stability

Ian Sellitto, Bertrand Le Bourdonnec, Karin Worm, Allan Goodman, Markku A. Savolainen, Guo-Hua Chu, Christopher W. Ajello, Christopher T. Saeui, Lara K. Leister, Joel A. Cassel, Robert N. DeHaven, Chr

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.40 MB

english, 2010

23

Design and Synthesis of Imidazopyrimidine Derivatives as Potent iNOS Dimerization Inhibitors

Chu, Guo-Hua, Le Bourdonnec, Bertrand, Gu, Minghua, Ajello, Christopher W, Leister, Lara K, Sellitto, Ian, Cassel, Joel A, Tuthill, Paul A, O’ Hare, Heather, DeHaven, Robert N, Dolle, Roland E

Journal:

The Open Medicinal Chemistry Journal

Year:

2009

File:

PDF, 746 KB

2009

24

Comparison of 3D Structures and AT 1 Binding Properties of Pyrazolidine-3,5-diones and Tetrahydropyridazine-3,6-diones with Parent Antihypertensive Drug Irbesartan

Le Bourdonnec, Bertrand, Cauvin, Christine, Meulon, Emmanuelle, Yous, Saïd, Goossens, Jean-François, Durant, François, Houssin, Raymond, Hénichart, Jean-Pierre

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 142 KB

english, 2002

25

Affinity labels as tools for the identification of opioid receptor recognition sites

Philip S Portoghese, Rachid El Kouhen, Ping Y Law, Horace H Loh, Bertrand Le Bourdonnec

Journal:

Year:

2001

Language:

english

File:

PDF, 165 KB

english, 2001

26

ChemInform Abstract: A New Synthesis of N-Alkyl Pyrazolidine-3,5-diones and Tetrahydropyridazine-3,6-diones.

Bertrand Le Bourdonnec, Emmanuelle Meulon, Said Yous, Raymond Houssin, Jean-Pierre Henichart

Journal:

Year:

2001

File:

PDF, 30 KB

2001

27

ChemInform Abstract: Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2009

Roland E. Dolle, Bertrand Le Bourdonnec, Karin Worm, Guillermo A. Morales, Craig J. Thomas, Wei Zhang

Journal:

Year:

2011

File:

PDF, 20 KB

2011

28

Synthesis and Pharmacological Evaluation of Novel Octahydro-1 H -pyrido[1,2-a]pyrazine as μ-Opioid Receptor Antagonists

Le Bourdonnec, Bertrand, Goodman, Allan J., Graczyk, Thomas M., Belanger, Serge, Seida, Pamela R., DeHaven, Robert N., Dolle, Roland E.

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 442 KB

english, 2006

29

The selective mu-opioid receptor antagonist adl5510 reduces levodopa-induced dyskinesia without affecting antiparkinsonian action in mptp-lesioned macaque model of Parkinson's disease

James B. Koprich, Susan H. Fox, Tom H. Johnston, Allan Goodman, Bertrand Le Bourdonnec, Roland E. Dolle, Robert N. DeHaven, Diane L. DeHaven-Hudkins, Patrick J. Little, Jonathan M. Brotchie

Journal:

Movement Disorders

Year:

2011

Language:

english

File:

PDF, 486 KB

english, 2011

30

General and efficient synthetic approach to novel tricyclic spiroketones

Guo-Hua Chu, Bertrand Le Bourdonnec, Minghua Gu, Christopher T. Saeui, Roland E. Dolle

Journal:

Year:

2009

Language:

english

File:

PDF, 266 KB

english, 2009

31

Reporter Affinity Labels: An o -Phthalaldehyde Derivative of β-Naltrexamine as a Fluorogenic Ligand for Opioid Receptors

Le Bourdonnec, Bertrand, El Kouhen, Rachid, Lunzer, Mary M., Law, Ping Y., Loh, Horace H., Portoghese, Philip S.

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 126 KB

english, 2000

32

CB2 selective sulfamoyl benzamides: Optimization of the amide functionality

Allan J. Goodman, Christopher W. Ajello, Karin Worm, Bertrand Le Bourdonnec, Markku A. Savolainen, Heather O’Hare, Joel A. Cassel, Gabriel J. Stabley, Robert N. DeHaven, Christopher J. LaBuda, Michael

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 494 KB

english, 2009

33

Novel trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidines as μ opioid receptor antagonists with improved opioid receptor selectivity profiles

Bertrand Le Bourdonnec, William M. Barker, Serge Belanger, Daniel D. Wiant, Nathalie C. Conway-James, Joel A. Cassel, Timothy J. O’Neill, Patrick J. Little, Robert N. DeHaven, Diane L. DeHaven-Hudkins

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 223 KB

english, 2008

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